PROTAC ERRalpha ligand 1, CAS [[1264754-13-3]]
Artikelnummer:
BYT-ORB1308355
Produktübersicht
Artikelname:
PROTAC ERRalpha ligand 1, CAS [[1264754-13-3]]
Artikelnummer:
BYT-ORB1308355
Hersteller Artikelnummer:
orb1308355
Alternativnummer:
BYT-ORB1308355-1,BYT-ORB1308355-10,BYT-ORB1308355-100,BYT-ORB1308355-2,BYT-ORB1308355-25,BYT-ORB1308355-5,BYT-ORB1308355-50,BYT-ORB1308355-500
Hersteller:
Biorbyt
Kategorie:
Biochemikalien
Alternative Synonym:
Inhibitor, ERR, ERRalpha, ERRgamma, Estrogen Receptor, EstrogenReceptor, Estrogen Receptor/ERR, inhibit, progestogen Receptor, progestogenReceptor, PROTAC ERRa ligand 1, PROTAC ERRalpha ligand 1, PROTAC ERRalpha ligand 1, PROTAC ERRalpha ligand1, PROTAC ERRalpha ligand-1
Produktbeschreibung
This compound is a potent and selective ERRalpha antagonist, with IC50 values of 0.04 µM for ERRalpha and 2.8 µM for ERRgamma. It serves as a key ligand for PROTAC development, enabling the targeted degradation of ERRalpha for research into its role in cancer, metabolism, and other cellular pathways in vitro.
Produkteigenschaften
Molekulargewicht:
420.36
Reinheit:
99.45% (May vary between batches)
CAS Nummer:
[1264754-13-3]
Formel:
C19H11F3N2O4S
Target-Kategorie:
Estrogen Receptor/ERR,Estrogen/progestogen Receptor
Anwendungsbeschreibung
Anwendungsbeschreibung:
Solubility: DMSO:120 mg/mL (285.47 mM),10% DMSO+40% PEG300+5% Tween 80+45% Saline:4 mg/mL (9.52 mM)