VU6028418 is a potent and selective orally bioavailable antagonist of the human M4 muscarinic acetylcholine receptor (hM4 mAChR), exhibiting an IC50 of 4.1 nM. This small molecule is a valuable research tool for investigating the role of M4 receptors in neurological disorders, supporting both in vitro binding studies and in vivo behavioral experiments.
Molekulargewicht:
432.491
CAS Nummer:
[2649803-05-2]
Formel:
C23H27F3N4O
Target-Kategorie:
AChR
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