NSC 12, CAS [[102586-30-1]]

Artikelnummer: BYT-ORB2813914
Artikelname: NSC 12, CAS [[102586-30-1]]
Artikelnummer: BYT-ORB2813914
Hersteller Artikelnummer: orb2813914
Alternativnummer: BYT-ORB2813914-1,BYT-ORB2813914-10,BYT-ORB2813914-25,BYT-ORB2813914-5,BYT-ORB2813914-50
Hersteller: Biorbyt
Kategorie: Biochemikalien
Alternative Synonym: NSC 12, NSC12, NSC-12
NSC 12 is an orally bioavailable pan-FGF inhibitor that traps FGF ligands, blocking FGFR1 signaling and disrupting tumor-promoting ternary complex formation without affecting heparin binding. It demonstrates antitumor activity by inhibiting cancer cell proliferation, angiogenesis, and metastasis in both cellular assays and animal models.
Molekulargewicht: 484.52
Reinheit: 99.51% (May vary between batches)
CAS Nummer: [102586-30-1]
Formel: C24H34F6O3
Target-Kategorie: FGFR
Anwendungsbeschreibung: Solubility: DMSO:8 mg/mL (16.51 mM),Ethanol:PBS (pH 7.2)(1:2):Insoluble,Ethanol:8 mg/mL (16.51 mM),DMF:8 mg/mL (16.51 mM)