MAK683 is a potent and selective small molecule inhibitor of the Embryonic Ectoderm Development (EED) protein, with IC50 values ranging from 26 to 89 nM across multiple biochemical assays. This inhibitor is a valuable chemical probe for investigating the role of EED and PRC2 complex function in epigenetic regulation, cancer biology, and stem cell research, both in vitro and in vivo.
Molekulargewicht:
376.39
Reinheit:
99.92% (May vary between batches)
CAS Nummer:
[1951408-58-4]
Formel:
C20H17FN6O
Target-Kategorie:
Histone Methyltransferase
Anwendungsbeschreibung:
Solubility: DMSO:4.33 mg/mL (11.5 mM)
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten